A facile synthesis of 1,4-diketones
- 作者Rolf Bergman; Bo Nilsson; Börje Wickberg
- 卷第31卷
- 期第19期
- 印刷ISSN0040-4039
- 文件大小231.69KB
- 发表时间1990
- DOI10.1016/s0040-4039(00)94698-7
- 页码2783-2786
Isolation and characterization of the duocarmycin-adenine DNA adductBoger, Dale L.; Ishizaki, Takayoshi; Zarrinmayeh, Hamideh · Journal of the American Chemical Society · 1991
(+)-CC-1065 DNA alkylation: observation of an unexpected relationship between cyclopropane electrophile reactivity and the intensity of DNA alkylationBoger, Dale L.; Munk, Stephen A.; Ishizaki, Takayoshi · Journal of the American Chemical Society · 1991
Synthesis and preliminary evaluation of agents incorporating the pharmacophore of the duocarmycin/pyrindamycin alkylation subunit: identification of the CC-1065/duocarmycin common pharmacophoreBoger, Dale L.; Ishizaki, Takayoshi; Zarrinmayeh, Hamideh; Kitos, P. A.; Suntornwat, O. · The Journal of Organic Chemistry · 1990
Duocarmycin-pyrindamycin DNA alkylation properties and identification, synthesis, and evaluation of agents incorporating the pharmacophore of the duocarmycin-pyrindamycin alkylation subunit. Identification of the CC-1065 duocarmycin common pharmacophoreBoger, Dale L.; Ishizaki, Takayoshi; Zarrinmayeh, Hamideh; Munk, Stephen A.; Kitos, Paul A.; Suntornwat, Oranart · Journal of the American Chemical Society · 1990
Synthesis of N-(phenylsulfonyl)-CI, N-((tert-butyloxy)carbonyl)-CI, CI-CDPI1, and CI-CDPI2: CC-1065 functional analog incorporating the parent 1,2,7,71-tetrahydrocycloprop[1,2-c]indol-4-one (CI) left-hand subunitBoger, Dale L.; Wysocki, Ronald J.; Ishizaki, Takayoshi · Journal of the American Chemical Society · 1990
Synthesis of N-(tert-butyloxycarbonyl)-CBI, CBI, CBI-CDPI1, and CBI-CDPI2: enhanced functional analogs of CC-1065 incorporating the 1,2,9,9a-tetrahydrocyclopropa[c]benz[e]indol-4-one (CBI) left-hand subunitBoger, Dale L.; Ishizaki, Takayoshi; Kitos, Paul A.; Suntornwat, Oranart · The Journal of Organic Chemistry · 1990
Total synthesis and evaluation of (.+-.)-N-(tert-butoxycarbonyl)-CBI, (.+-.)-CBI-CDPI1, and (.+-.)-CBI-CDPI2: CC-1065 functional agents incorporating the equivalent 1,2,9,9a-tetrahydrocyclopropa[1,2-c]benz[1,2-e]indol-4-one (CBI) left-hand subunitBoger, Dale L.; Ishizaki, Takayoshi; Wysocki, Ronald J.; Munk, Stephen A.; Kitos, Paul A.; Suntornwat, Oranart · Journal of the American Chemical Society · 1989