Pyrazolo[1,5-a]pyrimidine CRF-1 receptor antagonists
- 作者David J. Wustrow; Thomas Capiris; Ronald Rubin; James A. Knobelsdorf; Hyacinth Akunne; M.Duff Davis; Robert MacKenzie; Thomas A. Pugsley; Kim T. Zoski; Thomas G. Heffner; Lawrence D. Wise
- 卷第8卷
- 期第16期
- 印刷ISSN0960-894X
- 文件大小204.94KB
- 发表时间1998
- DOI10.1016/s0960-894x(98)00372-2
- 页码2067-2070
Peptidyl human heart chymase inhibitors. 1. Synthesis and inhibitory activity of difluoromethylene ketone derivatives bearing P′ binding subsitesMasahiro Eda; Atsuyuki Ashimori; Fumihiko Akahoshi; Takuya Yoshimura; Yoshihisa Inoue; Chikara Fukaya; Masahide Nakajima; Hajime Fukuyama; Teruaki Imada; Norifumi Nakamura · 1998
Peptidyl human heart chymase inhibitors. 2. Discovery of highly selective difluoromethylene ketone derivatives with Glu AT P3 siteMasahiro Eda; Atsuyuki Ashimori; Fumihiko Akahoshi; Takuya Yoshimura; Yoshihisa Inoue; Chikara Fukaya; Masahide Nakajima; Hajime Fukuyama; Teruaki Imada; Norifumi Nakamura · 1998
Corrigendum to “Peptidyl human heart chymase inhibitors. Part 1: Synthesis and inhibitory activity of difluoromethylene ketone derivatives bearing P′ binding subsites” [Bioorg. Med. Chem. Lett. 8 (1998) 913]Masahiro Eda; Atsuyuki Ashimori; Fumihiko Akahoshi; Takuya Yoshimura; Yoshihisa Inoue; Chikara Fukaya; Masahide Nakajima; Hajime Fukuyama; Teruaki Imada; Norifumi Nakamura · 1998