海量图书期刊资源,随时随地畅享阅读乐趣
Cancer: A drug-resistant duoLavoie, Hugo; Therrien, Marc · Nature · 2011
Regulation of RAF protein kinases in ERK signallingLavoie, Hugo; Therrien, Marc · Nature Reviews Molecular Cell Biology · 2015
Dimerization-induced allostery in protein kinase regulationLavoie, Hugo; Li, John J.; Thevakumaran, Neroshan; Therrien, Marc; Sicheri, Frank · Trends in Biochemical Sciences · 2014
MEK drives BRAF activation through allosteric control of KSR proteinsLavoie, Hugo; Sahmi, Malha; Maisonneuve, Pierre; Marullo, Sara A.; Thevakumaran, Neroshan; Jin, Ting; Kurinov, Igor; Sicheri, Frank; Therrien, Marc · Nature · 2018
RAF inhibitors promote RAS-RAF interaction by allosterically disrupting RAF autoinhibitionJin, Ting; Lavoie, Hugo; Sahmi, Malha; David, Maud; Hilt, Christine; Hammell, Amy; Therrien, Marc · Nature Communications · 2017
Time-resolved Phosphoproteome Analysis of Paradoxical RAF Activation Reveals Novel Targets of ERKKubiniok, Peter; Lavoie, Hugo; Therrien, Marc; Thibault, Pierre · Molecular & Cellular Proteomics · 2017
Crystal structure of a BRAF kinase domain monomer explains basis for allosteric regulationThevakumaran, Neroshan; Lavoie, Hugo; Critton, David A; Tebben, Andrew; Marinier, Anne; Sicheri, Frank; Therrien, Marc · Nature Structural & Molecular Biology · 2014