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Discovery of novel 2-(aminoheteroaryl)-thiazole-5-carboxamides as potent and orally active Src-family kinase p56Lck inhibitors

Discovery of novel 2-(aminoheteroaryl)-thiazole-5-carboxamides as potent and orally active Src-family kinase p56Lck inhibitors

Ping Chen; Derek Norris; Jagabandhu Das; Steven H. Spergel; John Wityak; Leslie Leith; Rulin Zhao; Bang-Chi Chen; Sidney Pitt; Suhong Pang; Ding Ren Shen; Rosemary Zhang; Henry F. De Fex; Arthur M. Doweyko; Kim W. McIntyre; David J. Shuster; Kamelia Behnia; Gary L. Schieven; Joel C. Barrish
  • 作者Ping Chen; Derek Norris; Jagabandhu Das; Steven H. Spergel; John Wityak; Leslie Leith; Rulin Zhao; Bang-Chi Chen; Sidney Pitt; Suhong Pang; Ding Ren Shen; Rosemary Zhang; Henry F. De Fex; Arthur M. Doweyko; Kim W. McIntyre; David J. Shuster; Kamelia Behnia; Gary L. Schieven; Joel C. Barrish
  • 卷第14卷
  • 期第24期
  • 印刷ISSN0960-894X
  • 文件大小351.75KB
  • 发表时间2004
  • DOI10.1016/j.bmcl.2004.09.093
  • 页码6061-6066
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