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Synthesis, initial SAR and biological evaluation of 1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-4-amine derived inhibitors of IκB kinase

Synthesis, initial SAR and biological evaluation of 1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-4-amine derived inhibitors of IκB kinase

James Kempson; Junqing Guo; Jagabandhu Das; Robert V. Moquin; Steven H. Spergel; Scott H. Watterson; Charles M. Langevine; Alaric J. Dyckman; Mark Pattoli; James R. Burke; XiaoXia Yang; Kathleen M. Gillooly; Kim W. McIntyre; Laishun Chen; John H. Dodd; Murray McKinnon; Joel C. Barrish; William J. Pitts
  • 作者James Kempson; Junqing Guo; Jagabandhu Das; Robert V. Moquin; Steven H. Spergel; Scott H. Watterson; Charles M. Langevine; Alaric J. Dyckman; Mark Pattoli; James R. Burke; XiaoXia Yang; Kathleen M. Gillooly; Kim W. McIntyre; Laishun Chen; John H. Dodd; Murray McKinnon; Joel C. Barrish; William J. Pitts
  • 卷第19卷
  • 期第10期
  • 印刷ISSN0960-894X
  • 文件大小1109.66KB
  • 发表时间2009
  • DOI10.1016/j.bmcl.2009.03.159
  • 页码2646-2649
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