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Design and optimization of a series of novel 2-cyano-pyrimidines as cathepsin K inhibitors

Design and optimization of a series of novel 2-cyano-pyrimidines as cathepsin K inhibitors

Zoran Rankovic; Jiaqiang Cai; Jennifer Kerr; Xavier Fradera; John Robinson; Ashvin Mistry; Emma Hamilton; George McGarry; Fiona Andrews; Wilson Caulfield; Iain Cumming; Maureen Dempster; John Waller; Paul Scullion; Iain Martin; Ann Mitchell; Clive Long; Mark Baugh; Paul Westwood; Emma Kinghorn; John Bruin; William Hamilton; Joost Uitdehaag; Mario van Zeeland; Dominique Potin; Laurent Saniere; Andre Fouquet; François Chevallier; Hortense Deronzier; Cecile Dorleans; Eric Nicolai
  • 作者Zoran Rankovic; Jiaqiang Cai; Jennifer Kerr; Xavier Fradera; John Robinson; Ashvin Mistry; Emma Hamilton; George McGarry; Fiona Andrews; Wilson Caulfield; Iain Cumming; Maureen Dempster; John Waller; Paul Scullion; Iain Martin; Ann Mitchell; Clive Long; Mark Baugh; Paul Westwood; Emma Kinghorn; John Bruin; William Hamilton; Joost Uitdehaag; Mario van Zeeland; Dominique Potin; Laurent Saniere; Andre Fouquet; François Chevallier; Hortense Deronzier; Cecile Dorleans; Eric Nicolai
  • 卷第20卷
  • 期第5期
  • 印刷ISSN0960-894X
  • 文件大小450.11KB
  • 发表时间2010
  • DOI10.1016/j.bmcl.2010.01.100
  • 页码1524-1527
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