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Design, synthesis and structure–activity relationships of (indo-3-yl) heterocyclic derivatives as agonists of the CB1 receptor. Discovery of a clinical candidate

Design, synthesis and structure–activity relationships of (indo-3-yl) heterocyclic derivatives as agonists of the CB1 receptor. Discovery of a clinical candidate

Paul Ratcliffe; Julia M. Adam; James Baker; Roberta Bursi; Robert Campbell; John K. Clark; Jean E. Cottney; Maureen Deehan; Anna-Marie Easson; Daniel Ecker; Darren Edwards; Ola Epemolu; Louise Evans; Ruth Fields; Stuart Francis; Paul Harradine; Fiona Jeremiah; Takao Kiyoi; Duncan McArthur; Angus Morrison; Paul Passier; Jack Pick; Peter G. Schnabel; Jurgen Schulz; Heinz Steinbrede; Glenn Walker; Paul Westwood; Grant Wishart; Joanna Udo de Haes
  • 作者Paul Ratcliffe; Julia M. Adam; James Baker; Roberta Bursi; Robert Campbell; John K. Clark; Jean E. Cottney; Maureen Deehan; Anna-Marie Easson; Daniel Ecker; Darren Edwards; Ola Epemolu; Louise Evans; Ruth Fields; Stuart Francis; Paul Harradine; Fiona Jeremiah; Takao Kiyoi; Duncan McArthur; Angus Morrison; Paul Passier; Jack Pick; Peter G. Schnabel; Jurgen Schulz; Heinz Steinbrede; Glenn Walker; Paul Westwood; Grant Wishart; Joanna Udo de Haes
  • 卷第21卷
  • 期第8期
  • 印刷ISSN0960-894X
  • 文件大小1364.25KB
  • 发表时间2011
  • DOI10.1016/j.bmcl.2011.02.023
  • 页码2541-2546
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