Identification of biaryl sulfone derivatives as antagonists of the histamine H3 receptor: Discovery of (R)-1-(2-(4′-(3-methoxypropylsulfonyl)biphenyl-4-yl)ethyl)-2-methylpyrrolidine (APD916)
Graeme Semple; Vincent J. Santora; Jeffrey M. Smith; Jonathan A. Covel; Rena Hayashi; Charlemagne Gallardo; Jason B. Ibarra; Jeffrey A. Schultz; Douglas M. Park; Scott A. Estrada; Brian J. Hofilena; Brian M. Smith; Albert Ren; Marissa Suarez; John Frazer; Jeffrey E. Edwards; Ryan Hart; Erin K. Hauser; Jodie Lorea; Andrew J. Grottick
- 作者Graeme Semple; Vincent J. Santora; Jeffrey M. Smith; Jonathan A. Covel; Rena Hayashi; Charlemagne Gallardo; Jason B. Ibarra; Jeffrey A. Schultz; Douglas M. Park; Scott A. Estrada; Brian J. Hofilena; Brian M. Smith; Albert Ren; Marissa Suarez; John Frazer; Jeffrey E. Edwards; Ryan Hart; Erin K. Hauser; Jodie Lorea; Andrew J. Grottick
- 卷第22卷
- 期第1期
- 印刷ISSN0960-894X
- 文件大小318.98KB
- 发表时间2012
- DOI10.1016/j.bmcl.2011.11.075
- 页码71-75