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Linker Immolation Determines Cell Killing Activity of Disulfide-Linked Pyrrolobenzodiazepine Antibody–Drug Conjugates

Linker Immolation Determines Cell Killing Activity of Disulfide-Linked Pyrrolobenzodiazepine Antibody–Drug Conjugates

Zhang, Donglu; Pillow, Thomas H.; Ma, Yong; Cruz-Chuh, Josefa dela; Kozak, Katherine R.; Sadowsky, Jack D.; Lewis Phillips, Gail D.; Guo, Jun; Darwish, Martine; Fan, Peter; Chen, Jingtian; He, Changrong; Wang, Tao; Yao, Hui; Xu, Zijin; Chen, Jinhua; Wai, John; Pei, Zhonghua; Hop, Cornelis E. C. A.; Khojasteh, S. Cyrus; Dragovich, Peter S.
  • 期刊名称ACS Medicinal Chemistry Letters
  • 作者Zhang, Donglu; Pillow, Thomas H.; Ma, Yong; Cruz-Chuh, Josefa dela; Kozak, Katherine R.; Sadowsky, Jack D.; Lewis Phillips, Gail D.; Guo, Jun; Darwish, Martine; Fan, Peter; Chen, Jingtian; He, Changrong; Wang, Tao; Yao, Hui; Xu, Zijin; Chen, Jinhua; Wai, John; Pei, Zhonghua; Hop, Cornelis E. C. A.; Khojasteh, S. Cyrus; Dragovich, Peter S.
  • 印刷ISSN1948-5875
  • 电子ISSN1948-5875
  • 文件大小1048.68KB
  • 发表时间2016-08-26
  • DOI10.1021/acsmedchemlett.6b00233
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