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Design, Synthesis and Characterization of Covalent KDM5 Inhibitors

Design, Synthesis and Characterization of Covalent KDM5 Inhibitors

Vazquez-Rodriguez, Saleta; Wright, Miranda; Rogers, Catherine M.; Cribbs, Adam; Velupillai, Srikannathasan; Philpott, Martin; Lee, Henry; Dunford, James E; Huber, Kilian V. M.; Robers, Mathew B.; Vasta, James D.; Thezenas, Marie Laetitia; Bonham, Sarah; Kessler, Benedikt; Bennett, James; Fedorov, Oleg; Raynaud, Florence; Donovan, Adam; Blagg, Julian; Bavetsias, Vassilios; Oppermann, Udo; Bountra, Chas; Kawamura, Akane; Brennan, Paul
  • 期刊名称Angewandte Chemie
  • 作者Vazquez-Rodriguez, Saleta; Wright, Miranda; Rogers, Catherine M.; Cribbs, Adam; Velupillai, Srikannathasan; Philpott, Martin; Lee, Henry; Dunford, James E; Huber, Kilian V. M.; Robers, Mathew B.; Vasta, James D.; Thezenas, Marie Laetitia; Bonham, Sarah; Kessler, Benedikt; Bennett, James; Fedorov, Oleg; Raynaud, Florence; Donovan, Adam; Blagg, Julian; Bavetsias, Vassilios; Oppermann, Udo; Bountra, Chas; Kawamura, Akane; Brennan, Paul
  • 印刷ISSN0044-8249
  • 文件大小1087.10KB
  • 发表时间2018-11-15
  • DOI10.1002/ange.201810179
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