Discovery and pharmacological evaluation of indole derivatives as potent and selective RORγt inverse agonist for multiple autoimmune conditions
Shaikh, Nadim S.; Iyer, Jitesh P.; Munot, Yogesh S.; Mukhopadhyay, Partha P.; Raje, Amol A.; Nagaraj, Ranganayaki; Jamdar, Vijay; Gavhane, Ravindra; Lohote, Mahendra; Sherkar, Prasad; Bala, Madhu; Petla, Rajkanth; Meru, Ashwinkumar; Umrani, Dhananjay; Rouduri, Sreekanth; Joshi, Sachin; Reddy, Satyanarayan; Kandikere, Vishwottam; Bhuniya, Debnath; Kulkarni, Bheemashankar; Mookhtiar, Kasim A.
- 期刊名称Bioorganic & Medicinal Chemistry Letters
- 作者Shaikh, Nadim S.; Iyer, Jitesh P.; Munot, Yogesh S.; Mukhopadhyay, Partha P.; Raje, Amol A.; Nagaraj, Ranganayaki; Jamdar, Vijay; Gavhane, Ravindra; Lohote, Mahendra; Sherkar, Prasad; Bala, Madhu; Petla, Rajkanth; Meru, Ashwinkumar; Umrani, Dhananjay; Rouduri, Sreekanth; Joshi, Sachin; Reddy, Satyanarayan; Kandikere, Vishwottam; Bhuniya, Debnath; Kulkarni, Bheemashankar; Mookhtiar, Kasim A.
- 印刷ISSN0960-894X
- 文件大小1593.62KB
- 发表时间2019-6
- DOI10.1016/j.bmcl.2019.06.044