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Discovery and pharmacological evaluation of indole derivatives as potent and selective RORγt inverse agonist for multiple autoimmune conditions

Discovery and pharmacological evaluation of indole derivatives as potent and selective RORγt inverse agonist for multiple autoimmune conditions

Shaikh, Nadim S.; Iyer, Jitesh P.; Munot, Yogesh S.; Mukhopadhyay, Partha P.; Raje, Amol A.; Nagaraj, Ranganayaki; Jamdar, Vijay; Gavhane, Ravindra; Lohote, Mahendra; Sherkar, Prasad; Bala, Madhu; Petla, Rajkanth; Meru, Ashwinkumar; Umrani, Dhananjay; Rouduri, Sreekanth; Joshi, Sachin; Reddy, Satyanarayan; Kandikere, Vishwottam; Bhuniya, Debnath; Kulkarni, Bheemashankar; Mookhtiar, Kasim A.
  • 期刊名称Bioorganic & Medicinal Chemistry Letters
  • 作者Shaikh, Nadim S.; Iyer, Jitesh P.; Munot, Yogesh S.; Mukhopadhyay, Partha P.; Raje, Amol A.; Nagaraj, Ranganayaki; Jamdar, Vijay; Gavhane, Ravindra; Lohote, Mahendra; Sherkar, Prasad; Bala, Madhu; Petla, Rajkanth; Meru, Ashwinkumar; Umrani, Dhananjay; Rouduri, Sreekanth; Joshi, Sachin; Reddy, Satyanarayan; Kandikere, Vishwottam; Bhuniya, Debnath; Kulkarni, Bheemashankar; Mookhtiar, Kasim A.
  • 印刷ISSN0960-894X
  • 文件大小1593.62KB
  • 发表时间2019-6
  • DOI10.1016/j.bmcl.2019.06.044
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