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A Phenotypic Screening Approach to Identify Anticancer Compounds Derived from Marine FungiEllinger, Bernhard; Silber, Johanna; Prashar, Anjali; Landskron, Johannes; Weber, Jonas; Rehermann, Sarah; Müller, Franz-Josef; Smith, Stephen; Wrigley, Stephen; Taskén, Kjetil; Gribbon, Philip; Labes, Antje; Imhoff, Johannes F. · ASSAY and Drug Development Technologies · 2014
Methoxylated 2'-hydroxychalcones as antiparasitic hit compoundsBorsari, Chiara; Santarem, Nuno; Torrado, Juan; Olías, Ana Isabel; Corral, María Jesús; Baptista, Catarina; Gul, Sheraz; Wolf, Markus; Kuzikov, Maria; Ellinger, Bernhard; Witt, Gesa; Gribbon, Philip; Reinshagen, Jeanette; Linciano, Pasquale; Tait, Annalisa; Costantino, Luca; Freitas-Junior, Lucio H.; Moraes, Carolina B.; Bruno dos Santos, Pascoalino; Alcântara, Laura Maria; Franco, Caio Haddad; Bertolacini, Claudia Danielli; Fontana, Vanessa; Tejera Nevado, Paloma; Clos, Joachim; Alunda, José María; Cordeiro-da-Silva, Anabela; Ferrari, Stefania; Costi, Maria Paola · European Journal of Medicinal Chemistry · 2017
Establishing the Secondary Metabolite Profile of the Marine Fungus: Tolypocladium geodes sp. MF458 and Subsequent Optimisation of Bioactive Secondary Metabolite ProductionKebede, Bethlehem; Wrigley, Stephen; Prashar, Anjali; Rahlff, Janina; Wolf, Markus; Reinshagen, Jeanette; Gribbon, Philip; Imhoff, Johannes; Silber, Johanna; Labes, Antje; Ellinger, Bernhard · Marine Drugs · 2017
EU-OPENSCREEN: A Novel Collaborative Approach to Facilitate Chemical BiologyBrennecke, Philip; Rasina, Dace; Aubi, Oscar; Herzog, Katja; Landskron, Johannes; Cautain, Bastien; Vicente, Francisca; Quintana, Jordi; Mestres, Jordi; Stechmann, Bahne; Ellinger, Bernhard; Brea, Jose; Kolanowski, Jacek L.; Pilarski, Radosław; Orzaez, Mar; Pineda-Lucena, Antonio; Laraia, Luca; Nami, Faranak; Zielenkiewicz, Piotr; Paruch, Kamil; Hansen, Espen; von Kries, Jens P.; Neuenschwander, Martin; Specker, Edgar; Bartunek, Petr; Simova, Sarka; Leśnikowski, Zbigniew; Krauss, Stefan; Lehtiö, Lari; Bilitewski, Ursula; Brönstrup, Mark; Taskén, Kjetil; Jirgensons, Aigars; Lickert, Heiko; Clausen, Mads H.; Andersen, Jeanette H.; Vicent, Maria J.; Genilloud, Olga; Martinez, Aurora; Nazaré, Marc; Fecke, Wolfgang; Gribbon, Philip · SLAS DISCOVERY: Advancing Life Sciences R&D · 2019
Profiling of flavonol derivatives for the development of anti-trypanosomatidic drugsBorsari, Chiara; Luciani, Rosaria; Pozzi, Cecilia; Pöhner, Ina; Henrich, Stefan; Trande, Matteo; Cordeiro-da-Silva, Anabela; Santarém, Nuno; Baptista, Catarina; Tait, Annalisa; Di Pisa, Flavio; Dello Iacono, Lucia; Landi, Giacomo; Gul, Sheraz; Wolf, Markus; Kuzikov, Maria; Ellinger, Bernhard; Reinshagen, Jeanette; Witt, Gesa; Gribbon, Philip; Kohler, Manfred; Keminer, Oliver; Behrens, Birte; Costantino, Luca; Tejera Nevado, Paloma; Bifeld, Eugenia; Eick, Julia; Clos, Joachim; Torrado, Juan; Jiménez-Antón, María Dolores; Corral, Maria Jesùs; Alunda, José Maria; Pellati, Federica; Wade, Rebecca C; Ferrari, Stefania; Mangani, Stefano; Costi, Maria Paola · Journal of Medicinal Chemistry · 2016
Exploiting the 2-Amino-1,3,4-thiadiazole Scaffold To Inhibit <i>Trypanosoma brucei</i> Pteridine Reductase in Support of Early-Stage Drug DiscoveryLinciano, Pasquale; Dawson, Alice; Pöhner, Ina; Costa, David M.; Sá, Monica S.; Cordeiro-da-Silva, Anabela; Luciani, Rosaria; Gul, Sheraz; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Gribbon, Philip; Reinshagen, Jeanette; Wolf, Markus; Behrens, Birte; Hannaert, Véronique; Michels, Paul A. M.; Nerini, Erika; Pozzi, Cecilia; di Pisa, Flavio; Landi, Giacomo; Santarem, Nuno; Ferrari, Stefania; Saxena, Puneet; Lazzari, Sandra; Cannazza, Giuseppe; Freitas-Junior, Lucio H.; Moraes, Carolina B.; Pascoalino, Bruno S.; Alcântara, Laura M.; Bertolacini, Claudia P.; Fontana, Vanessa; Wittig, Ulrike; Müller, Wolfgang; Wade, Rebecca C.; Hunter, William N.; Mangani, Stefano; Costantino, Luca; Costi, Maria P. · ACS Omega · 2017
<b>Network approaches to drug discovery</b>Chandra, Nagasuma; Padiadpu, Jyothi · Expert Opinion on Drug Discovery · 2013
Animal models of anorexia and cachexiaDeBoer, Mark D · Expert Opinion on Drug Discovery · 2009
Contextual data integration in drug discoveryYuryev, Anton · Expert Opinion on Drug Discovery · 2012
The antibiotic resistomeWright, Gerard D · Expert Opinion on Drug Discovery · 2010
Leadhopping – and beyondCramer, Richard D · Expert Opinion on Drug Discovery · 2006
Descriptors for antimicrobial peptidesJenssen, Håvard · Expert Opinion on Drug Discovery · 2011
Preclinical development of therapeutic biologicsBaumann, Andreas · Expert Opinion on Drug Discovery · 2008
Ayurvedic drug discoveryBalachandran, Premalatha; Govindarajan, Rajgopal · Expert Opinion on Drug Discovery · 2007